Pentamidine: Side Effects, Uses & Monitoring

Facts extracted from current FDA product labeling for Pentamidine. Educational only — not medical advice.

Reported adverse reactions

ReactionHighest frequency reported*
Impaired renal function28.8%
Elevated serum creatinine23.6%
Leukopenia10.4%
Elevated liver function tests8.7%
Azotemia8.5%
Elevated blood urea nitrogen6.6%
Anorexia/nausea5.9%
Hypoglycemia5.9%
Hypotension5%
Rash3.3%
Thrombocytopenia2.6%
Confusion/hallucinations1.7%
Bad taste1.7%
Anemia1.2%

*Highest percentage across placebo-controlled trial tables summarized in current labeling.

Labeled uses

Pentamidine isethionate for injection is indicated for the treatment of pneumonia due to Pneumocystis carinii .

Source: FDA labeling via NIH DailyMed (set 860c799c…). Not affiliated with FDA or NIH.

Medical disclaimer: Always consult a qualified healthcare professional about any medication.