Leuprolide: Side Effects, Uses & Monitoring

Facts extracted from current FDA product labeling for Leuprolide. Educational only — not medical advice.

Reported adverse reactions

ReactionHighest frequency reported*
Gynecomastia/breast tenderness or pain63%
Hot flashes55%
Peripheral edema30%
Ecg changes/ischemia22%
Nausea/vomiting17%
General pain13%
Impotence12%
Phlebitis/thrombosis10%
Asthenia10%
Constipation9%
Myalgia9%
High blood pressure8%
Murmur8%
Dyspnea8%
Dermatitis8%
Frequency/urgency8%
Dizziness/lightheadedness7%
Headache7%
Insomnia/sleep disorders7%
Urinary tract infection7%

*Highest percentage across placebo-controlled trial tables summarized in current labeling.

Labeled uses

Leuprolide acetate injection is indicated in the palliative treatment of advanced prostatic cancer.

Source: FDA labeling via NIH DailyMed (set a3b01473…). Not affiliated with FDA or NIH.

Medical disclaimer: Always consult a qualified healthcare professional about any medication.